Description

(Liquid Formulation of PDE5 Inhibitor for Erectile Dysfunction and Vascular Support)

Flexible, Fast-Acting Alternative to Oral Tablets for Sexual Health and Vasodilation Therapy

Sildenafil Drops offer a liquid, titratable formulation of the well-known PDE5 inhibitor used to treat erectile dysfunction (ED), as well as select off-label vascular conditions. Each 30 mL bottle contains a total of 100 mg of sildenafil citrate, delivered in a drop-based dosing format that allows for precise micro-dosing, rapid absorption, and convenient administration—especially for individuals who prefer not to take tablets or who require flexible titration.

Compounded by prescription, this formulation is ideal for patients seeking a customized dosing solution to support sexual performance, vascular responsiveness, and in some cases, exercise tolerance or pulmonary vascular conditions under clinical supervision.

Product Overview

• Active Ingredient: Sildenafil Citrate

• Concentration: 100 mg total per 30 mL

• Form: Oral liquid (drop formulation)

• Delivery: By dropper or measured syringe

• Use: Erectile dysfunction, vascular enhancement, off-label support for pulmonary conditions

• Storage: Room temperature (20–25°C); refrigerate if directed

• Packaging: Amber 30 mL dropper bottle

• Availability: Prescription-only; compounded formulation

What Is Sildenafil?

Sildenafil is a phosphodiesterase type 5 (PDE5) inhibitor that works by enhancing the effects of nitric oxide, a natural vasodilator, in vascular smooth muscle. It is most widely used to:

• Treat erectile dysfunction (ED) in men

• Support sexual arousal response via increased penile blood flow

• Improve endothelial function and vascular tone in specific medical conditions

The drop-based formulation provides a non-tablet alternative, allowing for more individualized and dynamic use, especially in patients with:

• Swallowing difficulties

• Need for flexible or partial dosing

• Preference for rapid titration with fewer side effects

Mechanism of Action

Sildenafil inhibits PDE5, an enzyme that breaks down cyclic guanosine monophosphate (cGMP). By increasing cGMP levels, sildenafil promotes:

• Relaxation of vascular smooth muscle

• Improved blood flow to the corpus cavernosum of the penis

• Enhanced erection quality, rigidity, and duration during sexual stimulation

• Lowered pulmonary vascular resistance (off-label applications)

This action requires sexual arousal to be effective and does not induce spontaneous erections.

Clinical Uses

1. Erectile Dysfunction (ED)

• Improves erection response to sexual stimulation

• Especially effective in men with mild-to-moderate ED, age-related vascular decline, or performance anxiety

• Allows dose customization based on sensitivity or side-effect profile

2. Vascular Support

• Off-label use in some protocols for pulmonary hypertension, Raynaud’s syndrome, or vascular insufficiency

• May aid in exercise performance in certain cardiac rehabilitation settings (by prescription only)

3. Sexual Wellness and Lifestyle Protocols

• Integrated into biohacking or anti-aging programs focused on vascular optimization and intimacy health

Dosing and Administration

• Typical ED Starting Dose: 5–20 mg (1.5–6 mL depending on compounding instructions) taken orally 30–60 minutes before sexual activity

• Max Frequency: Once per 24 hours

• Adjustment: May be increased or decreased based on efficacy and tolerability

• Administration: Use calibrated dropper or oral syringe for accurate measurement

Always follow compounding pharmacy or prescriber-specific instructions, as concentration may vary slightly by batch.

Safety and Tolerability

Sildenafil is well tolerated, especially in liquid form where smaller doses can be administered and titrated.

Common mild side effects include:

• Headache

• Flushing

• Nasal congestion

• Indigestion

• Visual disturbances (blue-tinged vision, light sensitivity)

These effects are dose-dependent and generally mild.

Serious Side Effects (Rare)

• Sudden vision or hearing loss

• Priapism (erection >4 hours)

• Hypotension when combined with nitrates or alpha-blockers

• Cardiovascular events in high-risk patients (rare with appropriate screening)

Contraindications

Do not use if:

• Taking nitrate medications (risk of severe hypotension)

• History of retinal disorders (e.g., NAION)

• Severe cardiovascular disease without physician approval

• Known allergy to sildenafil or similar compounds

Use caution in patients with liver/kidney disease or those on multiple antihypertensives.

Storage and Handling

• Store in a cool, dry place (room temperature or as labeled)

• Shake well before each use if suspension-based

• Keep dropper clean and tightly sealed

• Use within 30–60 days of opening or per pharmacy guidance

• Keep out of reach of children

Why Choose Sildenafil Drops?

• Allows for microdosing and flexible titration

• Faster absorption and onset than traditional tablets for some users

• Easier administration for those with pill aversion or dysphagia

• Supports personalized ED therapy or off-label vascular care

• Custom-compounded for purity and consistent concentration

Summary

Sildenafil Drops – 100 mg in 30 mL Oral Liquid provide a convenient, precisely dosed alternative to traditional ED medications. Whether used to manage erectile dysfunction, support vascular function, or enhance sexual wellness, this formulation offers flexibility, discretion, and clinical-grade reliability. Custom-compounded for safety and absorption, it’s an ideal option for patients seeking personalized performance enhancement under medical guidance.