Description

(Selective Growth Hormone Secretagogue for Anti-Aging, Recovery, and Body Composition)

A Targeted Approach to Growth Hormone Optimization Without Unwanted Side Effects

Ipamorelin is a highly selective growth hormone secretagogue (GHS) that stimulates the natural release of growth hormone (GH) from the anterior pituitary gland, without significantly affecting cortisol, prolactin, or appetite. This pharmaceutical-grade formulation provides 15 mg of lyophilized Ipamorelin in a single-use vial, intended for reconstitution with 5 mL bacteriostatic water, yielding a 3 mg/mL concentration for subcutaneous or intramuscular injection under medical supervision.

Favored in anti-aging medicine, hormone optimization, fitness recovery, and functional wellness, Ipamorelin has become one of the most trusted GH-releasing peptides due to its clean profile, minimal side effects, and natural mimicry of the body’s growth hormone pulse.

Product Overview

• Active Ingredient: Ipamorelin acetate
• Dosage Form: Lyophilized powder
• Total Peptide Content: 15 mg per vial
• Reconstitution Volume: 5 mL bacteriostatic water (final concentration: 3 mg/mL)
• Administration: Subcutaneous or intramuscular injection
• Storage (Unmixed): 2–8°C (36–46°F)
• Storage (After Reconstitution): Refrigerate and use within 30 days
• Use: Physician-supervised peptide therapy

What Is Ipamorelin?

Ipamorelin is a synthetic pentapeptide developed to replicate the function of ghrelin at the growth hormone secretagogue receptor (GHS-R1a). It is part of the newer class of peptides that stimulate endogenous GH release while avoiding the unwanted stimulation of cortisol, aldosterone, prolactin, or intense hunger—effects commonly seen with earlier GHRPs like GHRP-6 and GHRP-2.

Its clean safety profile and specificity for growth hormone secretion make it a well-tolerated and effective option for adults seeking:

• Enhanced recovery and healing
• Improved body composition
• Hormonal rejuvenation
• Anti-aging support

Mechanism of Action

Ipamorelin binds to ghrelin receptors in the hypothalamus and pituitary gland to stimulate natural GH release. It enhances the body’s physiological growth hormone pulses while preserving the body’s negative feedback loop, which helps prevent overstimulation.

Key benefits include:

• Stimulation of GH release without increasing cortisol or prolactin
• Support for lean muscle development and fat loss
• Improved tissue repair, sleep, and metabolic regulation
• Promotion of collagen synthesis and skin health
• Enhanced cellular regeneration and cognitive function

Clinical Applications

Ipamorelin is widely used in:

1. Hormone Optimization and Anti-Aging

• Supports natural GH and IGF-1 levels
• Reduces signs of aging (skin laxity, poor recovery, energy decline)
• Helps mitigate age-related muscle loss (sarcopenia)

2. Recovery and Healing

• Speeds up post-surgical and post-injury repair
• Improves tendon and joint recovery
• Beneficial for athletes and active individuals under strain

3. Body Composition

• Promotes fat metabolism and muscle preservation
• Enhances protein synthesis
• Improves metabolic flexibility and endurance

4. Sleep and Cognitive Function

• Improves deep sleep and GH-dependent circadian balance
• May enhance mood, clarity, and focus due to hormonal balance

Dosing and Administration

• Typical dose: 200–300 mcg once or twice daily
• Timing: Best administered on an empty stomach, ideally post-workout or before bedtime
• Route: Subcutaneous injection in abdominal or thigh region
• Cycle Length: 8–12 weeks with optional 2–4 week break

Reconstitution instructions: Use 5 mL bacteriostatic water. Swirl gently—do not shake.

Safety and Side Effects

Ipamorelin has one of the best safety profiles among GH secretagogues. It is well-tolerated and typically free from the adverse effects associated with older GHRPs.

Mild potential effects may include:

• Temporary injection site redness
• Lightheadedness or flushing (rare)
• Mild water retention in some users
• Tingling or slight numbness in extremities (related to GH elevation)

It does not increase cortisol, prolactin, or hunger, making it ideal for long-term, balanced use.

Contraindications and Cautions

Do not use if:

• You are pregnant or breastfeeding
• You have active cancer or growth hormone-sensitive tumors
• You are taking medications with GH-interfering properties without provider oversight

Caution advised in individuals with untreated thyroid, adrenal, or pituitary conditions.

Storage and Handling

• Before reconstitution: Store at 2–8°C
• After reconstitution: Keep refrigerated and use within 30 days
• Use sterile technique to prevent contamination
• Do not freeze; avoid repeated temperature cycling

Why Choose Ipamorelin?

• Highly selective and safe GH stimulation
• No significant appetite increase or hormonal imbalance
• Compatible with other peptide therapies (e.g., CJC-1295)
• Promotes gradual, sustainable results
• Trusted in anti-aging, wellness, and performance practices

Summary

Ipamorelin – 15 mg Vial (Reconstituted to 5 mL at 3 mg/mL) offers a refined, effective, and well-tolerated strategy for boosting natural growth hormone production, improving body composition, and supporting recovery, sleep, and healthy aging. Whether as part of an integrated longevity plan or targeted recovery protocol, Ipamorelin delivers reliable performance with minimal side effects, making it a cornerstone of modern peptide-based hormone support.